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Search Results for " g-protein coupled receptor 1 "
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Targets

63

Compounds

5

Natural Products

1749

Recombinant Proteins

1

Libraries

Cat No. Product Name Synonyms Targets
T7428 SBI-115 GPCR19
SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5
T4083 BAR501 BAR 501 GPCR19
BAR501 is an effective and specific GPBAR1 agonist (EC50: 1 μM).
TQ0252 BAR502 FXR , GPCR19 , Autophagy
BAR502 is a dual GPBAR1 and FXR agonist (IC50s: 0.4 μM and 2 μM).
T4352 SB756050 SB-756050,SB 756050 GPCR19
SB756050 is a specific TGR5 agonist.
T8818 TC-G 1005 GPCR19
TC-G 1005 is a potent and selective GPBA agonist (EC50 :0.72 nM; hTGR5). Selective for TGR5 over FXR (farnesoid X receptor). Increases plasma GLP-1 levels and reduces blood glucose in mice. Orally available.
T1824 TGR5 Receptor Agonist GPCR19
TGR5 is a potent TGR5(GPCR19) agonist.
T36036 CAY10786 GPR52 antagonist-1 GPR
CAY10786 (GPR52 antagonist-1) is an antagonist of G protein-coupled receptor 52 (GPR52, IC50 = 0.63 μM).
T12104 MRGPRX1 agonist 1 Others
MRGPRX1 agonist 1 is a highly potent MRGPRX1 (Mas-related G-protein-coupled receptor X1)agonist(EC50 of 50 nM).
T3498 CCG215022 GRK , PKA
CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.
T7847 Apelin-13 triTFA(217082-58-1(free base)) Others
Apelin-13 triTFA is the endogenous ligand of the APJ receptor, activating this G protein-coupled receptor with an EC50 value of 0.37 nM.
TP1982L Neuropeptide S (Rat) acetate Neuropeptide Y Receptor
Neuropeptide S (Rat) acetate is an endogenous ligand of a previously orphan G-protein-coupled receptor now named NPS receptor. Neuropeptide S (Rat) acetate can be used for the research of nervous system disease [1].
T60199 NCRW0005-F05 GPR
NCRW0005-F05 is a potent agonist of orphan G-protein coupled receptor GPR139 with an IC 50 value of 0.21 μM. NCRW0005-F05 can be used to research diabetes, obesity and Parkinson's disease [1].
T63166 LSN3318839 LSN-3318839,LSN 3318839 Glucagon Receptor
LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can be used to lower blood glucose.
TP2296L TLQP 21 acetate Complement System
TLQP 21 acetate is a potent agonist of G-protein-coupled receptor complement-3a receptor 1 (C3aR1). The EC50 values are 10.3 μM for mouse and 68.8 μM for human. TLQP 21 acetate is a VGF-derived peptide with endocrine a...
T37496L Alamandine TFA RAAS
Alamandine TFA , a member of the renin-angiotensin system (RAS), a vasoactive peptide, is an endogenous ligand of the G protein-coupled receptor MrgD. Alamandine TFA targets to protect the kidney and heart through anti-h...
T15810 LY2922470 GPR
LY2922470 reduces glucose levels along with significant enhancements in insulin and GLP-1, which is the potential for the treatment of type 2 diabetes mellitus (T2DM). LY2922470 is an effective, selective, and orally ava...
T38287 C3a Receptor Agonist C3a receptor agonist 1,Complement 3a Receptor Agonist Complement System
C3a Receptor Agonist (C3a receptor agonist 1) binds the G protein-coupled C3a receptors (C3aRs) in the immune system complement pathway. Activation of C3aR prevents neutrophils from being mobilized in a model of intestin...
T13714 CCG258208 GRK2-IN-1 GRK
GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).
T40517 GPR30 agonist-1 GPR30 agonist-1
GPR30 agonist-1 is a compound that acts as an agonist for G protein-coupled receptor 30 (GPR30), inducing vasorelaxation.
T82265 GPR3 agonist-2
GPR3 agonist-2 (compound 32) is a potent full agonist of the G protein-coupled receptor 3 (GPR3), exhibiting an IC50 value of 260 nM [1].
T35875 CCG258208 hydrochloride
GRKs-IN-1 hydrochloride, Compound 14as, has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50=130 nM) and GRK5 (IC50=7.1 μM).GRKs-IN-1 hydrochloride is a derivative 14as of pa...
T13714L GRK2-IN-1 hydrochloride (2055990-90-2 free base) GRK2-IN-1 hydrochloride GRK
GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).
T82258 GRL018-21
GRL018-21 is a potent, highly selective inhibitor of G protein-coupled receptor kinase 5 (GRK5), exhibiting an IC50 of 10 nM [1].
T12744 RO5256390 Others
RO5256390 is a trace amine-associated receptor 1 (TAAR1) agonist, a highly conserved G-protein-coupled receptor that blocks psychostimulant-induced hyperarousal, and may be used in the study of neurological disorders.
T76423 Neuropeptide AF (cattle)
Neuropeptide AF (cattle), an amidated octadecapeptide and RFamide neuropeptide, serves as a ligand for Mas-related gene receptor A4 (MrgprA4) (Mas-related G-protein-coupled Receptor (MRGPR)) with an EC50 of approximately...
T83547 (Des-Bromo)-Neuropeptide B (1-23) (human)
'(Des-Bromo)-Neuropeptide B (1-23) (human)' is an agonist for orphan G-protein-coupled receptors, exhibiting a K i of 1.2 nM for GPR7 (NPBW1) and 341 nM for GPR8 (NPBW2) respectively [1].
T60497 MRGPRX1 agonist 3
MRGPRX1 agonist 3 (compound 1f) is a potent positive allosteric modulator of Mas-related G protein-coupled receptor X1 (MRGPRX1) with an EC50 of 0.22 μM. MRGPRX1 agonist 3 can be used for neuropathic pain research[1].
T75962 Urotensin II, mouse acetate
Urotensin II, mouse acetate, serves as an endogenous ligand for the orphan G-protein-coupled receptor GPR14 or SENR and acts as a potent vasoconstrictor. Its physiological function extends to the central nervous system [...
T75961 Urotensin II, mouse TFA
Urotensin II, mouse TFA, an endogenous ligand for the orphan G-protein-coupled receptor GPR14 or SENR, serves as a potent vasoconstrictor. It plays a significant physiological role within the central nervous system [1].
T81683 Neuromedin S (human)
Neuromedin S (human) is a 33-amino acid neuropeptide identified as an endogenous ligand for the orphan G-protein coupled receptor (GPCR) FM-4/TGR-1, acting on the neuromedin U (NMU) receptor 2 (NMUR2) to regulate body we...
T38077 TLQP-21 TFA
TLQP-21 TFA, a VGF-derived peptide endowed of endocrine and extraendocrine properties, is a potent G-protein-coupled receptor complement-3a receptor1 (C3aR1) agonist (EC50: mouse TLQP-21=10.3 μM; human TLQP-21=68.8μM). T...
T63554 TGR5 Receptor Agonist 3
TGR5 Receptor Agonist 3 is a G protein-coupled bile acid receptor 1 (GPBAR1, TGR5) agonist soft drug compound that decreases gallbladder filling, exhibits good gallbladder safety, and is able to act on hTGR5 (EC50: 16.4 ...
T70468 MK-8666
MK-8666 is a partial GPCR (G-protein-coupled receptor) agonist that is coordinated with the action of GPR40. GPR40, also known as free fatty acid (FFA) receptor 1 modulates fatty acid-induced insulin secretion in pancrea...
T62518 GRK6-IN-1
GRK6-IN-1 (compound 18) is a potent inhibitor of G protein-coupled receptor kinase 6 (GRK6) (IC50: 120 nM). GRK6-IN-1 has the potential to be studied in multiple myeloma.
T81682 Neuromedin S(rat) TFA
Neuromedin S(rat) TFA, a 34-amino acid peptide derivative of rat Neuromedin S, is a neuropeptide sourced from the rat brain that functions as a ligand for the G protein-coupled receptor FM4/TGR-1 [1].
T60466 MRGPRX1 agonist 2
MRGPRX1 agonist 2 (compound 1a) is a potent positive allosteric modulator of Mas-related G protein-coupled receptor X1 (MRGPRX1) with an EC 50 value of 0.48 μM. MRGPRX1 agonist 2 has the potential to be used in neuropath...
T69953 MK-8666 Tris
MK-8666 Tris is a partial GPCR (G-protein-coupled receptor) agonist that is coordinated with the action of GPR40. GPR40, also known as free fatty acid (FFA) receptor 1 modulates fatty acid-induced insulin secretion in pa...
T37303 5-OxoETE 5-KETE,5-OxoETE
5-OxoETE is a polyunsaturated keto acid formed by the oxidation of 5-HETE in human neutrophils by a specific dehydrogenase.[1] It stimulates cytosolic calcium levels in neutrophils with an EC50 value of 2 nM.[2] 5-OxoETE...
T62918 GPR84 antagonist 3
GPR84 Antagonist 3 (compound 42), a potent inhibitor of the G-protein-coupled receptor 84 (GPR84), exhibits a pIC50 value of 8.28, indicating strong antagonistic activity by inhibiting GTPγS. Additionally, it possesses a...
T35839 3-Iodothyronamine (hydrochloride)
3-Iodothyronamine is derived from the deiodination and decarboxylation of endogenous thyroxine. It activates the G protein-coupled receptor known as trace amine-associated receptor 1 at nanomolar concentrations whereupon...
T36080 Rivenprost ONO-4819
Prostaglandin E2 activates four distinct G protein-coupled receptors, EP1-4. Rivenprost is a potent and selective agonist for the EP4 receptor (Ki = 0.7, 56, 620, and >10,000 nM for EP4, EP3, EP2, and EP1, respectively)....
T76262 Cagrilintide
Cagrilintide, an investigational novel long-acting acylated amylin analogue, functions as an agonist for nonselective amylin receptors (AMYR) and the calcitonin G protein-coupled receptor (CTR). It significantly reduces ...
T75784 Apelin-36(rat, mouse) TFA
Apelin-36(rat, mouse) TFA, an endogenous agonist for the orphan G protein-coupled receptor APJ, exhibits a strong affinity for APJ receptors with an IC 50 of 5.4 nM and effectively inhibits cAMP production with an EC 50 ...
T36982 CXCR3 Antagonist 6c
CXCR3 antagonist 6c is an antagonist of chemokine (C-X-C motif) receptor 3 (CXCR3).1It inhibits calcium mobilization induced by chemokine (C-X-C motif) ligand 11 (CXCL11) in HEK293 cells expressing the human receptor (IC...
T75785 Apelin-17(human, bovine) TFA
Apelin-17(human, bovine) TFA is an endogenous agonist of the orphan G protein-coupled receptor APJ. This compound demonstrates affinity for human APJ receptors on HEK 293 cells, evidenced by a pIC50 value of 9.02. Additi...
T35855 AAA
AAA is an antagonist of G protein-coupled receptor 75 (GPR75).1It increases basal GPR75 protein levels and inhibits 20-HETE-induced reductions in GPR75 protein levels in PC3 cells. AAA (5 and 10 μM) also reduces 20-HETE-...
T71338 Patidegib HCl
Patidegip, laos known as Saridegib and IPI-926, is an orally bioavailable, cyclopamine-derived (for structure comparison see Fig 1) inhibitor of the Hedgehog (Hh) pathway with potential antineoplastic activity. Specific...
T75901 Obestatin(rat) TFA
Obestatin(rat) TFA is a cpeptide derived from the Ghrelin gene, consisting of 23 amino acids. This compound modulates physiological processes by suppressing food intake, inhibiting jejunal contraction, and reducing body-...
T38336 W140 (trifluoroacetate salt) W140 (trifluoroacetate salt)
Sphingosine-1-phosphate (S1P) is a bioactive lipid that exhibits a broad spectrum of biological activities including cell proliferation, survival, migration, cytoskeletal organization, and morphogenesis. It exerts its ac...
T75925 Orexin B, rat, mouse TFA
Orexin B, rat, mouse (Rat orexin B) TFA, an endogenous agonist for orexin receptors, binds to and activates the closely related orphan G protein-coupled receptors OX1-R and OX2-R. This compound is instrumental in stimula...

Compounds

SBI-115
T7428
Synonym:
Target: GPCR19
BAR501
T4083
Synonym: BAR 501
Target: GPCR19
BAR502
TQ0252
Synonym:
Target: FXR, GPCR19, Autophagy
SB756050
T4352
Synonym: SB-756050,SB 756050
Target: GPCR19
TC-G 1005
T8818
Synonym:
Target: GPCR19
TGR5 Receptor Agonist
T1824
Synonym:
Target: GPCR19
CAY10786
T36036
Synonym: GPR52 antagonist-1
Target: GPR
MRGPRX1 agonist 1
T12104
Synonym:
Target: Others
CCG215022
T3498
Synonym:
Target: GRK, PKA
Apelin-13 triTFA(217082-58-1(free base))
T7847
Synonym:
Target: Others
Neuropeptide S (Rat) acetate
TP1982L
Synonym:
Target: Neuropeptide Y Receptor
NCRW0005-F05
T60199
Synonym:
Target: GPR
LSN3318839
T63166
Synonym: LSN-3318839,LSN 3318839
Target: Glucagon Receptor
TLQP 21 acetate
TP2296L
Synonym:
Target: Complement System
Alamandine TFA
T37496L
Synonym:
Target: RAAS
LY2922470
T15810
Synonym:
Target: GPR
C3a Receptor Agonist
T38287
Synonym: C3a receptor agonist 1,Complement 3a Receptor Agonist
Target: Complement System
CCG258208
T13714
Synonym: GRK2-IN-1
Target: GRK
GPR30 agonist-1
T40517
Synonym: GPR30 agonist-1
Target:
GPR3 agonist-2
T82265
Synonym:
Target:
CCG258208 hydrochloride
T35875
Synonym:
Target:
GRK2-IN-1 hydrochloride (2055990-90-2 free base)
T13714L
Synonym: GRK2-IN-1 hydrochloride
Target: GRK
GRL018-21
T82258
Synonym:
Target:
RO5256390
T12744
Synonym:
Target: Others
Neuropeptide AF (cattle)
T76423
Synonym:
Target:
(Des-Bromo)-Neuropeptide B (1-23) (human)
T83547
Synonym:
Target:
MRGPRX1 agonist 3
T60497
Synonym:
Target:
Urotensin II, mouse acetate
T75962
Synonym:
Target:
Urotensin II, mouse TFA
T75961
Synonym:
Target:
Neuromedin S (human)
T81683
Synonym:
Target:
TLQP-21 TFA
T38077
Synonym:
Target:
TGR5 Receptor Agonist 3
T63554
Synonym:
Target:
MK-8666
T70468
Synonym:
Target:
GRK6-IN-1
T62518
Synonym:
Target:
Neuromedin S(rat) TFA
T81682
Synonym:
Target:
MRGPRX1 agonist 2
T60466
Synonym:
Target:
MK-8666 Tris
T69953
Synonym:
Target:
5-OxoETE
T37303
Synonym: 5-KETE,5-OxoETE
Target:
GPR84 antagonist 3
T62918
Synonym:
Target:
3-Iodothyronamine (hydrochloride)
T35839
Synonym:
Target:
Rivenprost
T36080
Synonym: ONO-4819
Target:
Cagrilintide
T76262
Synonym:
Target:
Apelin-36(rat, mouse) TFA
T75784
Synonym:
Target:
CXCR3 Antagonist 6c
T36982
Synonym:
Target:
Apelin-17(human, bovine) TFA
T75785
Synonym:
Target:
AAA
T35855
Synonym:
Target:
Patidegib HCl
T71338
Synonym:
Target:
Obestatin(rat) TFA
T75901
Synonym:
Target:
W140 (trifluoroacetate salt)
T38336
Synonym: W140 (trifluoroacetate salt)
Target:
Orexin B, rat, mouse TFA
T75925
Synonym:
Target:
1 2
Cat No. Product Name Synonyms Targets
T5077 Deoxycholic acid sodium salt Sodium deoxycholate,Sodium Desoxycholate Endogenous Metabolite , GPCR19
Deoxycholic acid sodium salt (Sodium deoxycholate) can activate the G protein-coupled bile acid receptor TGR5 that stimulates brown adipose tissue (BAT) thermogenic activity.
T2965 Deoxycholic acid Cholorebic,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic Endogenous Metabolite , GPCR19
Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate. It is usually conjugated with glycine or taurine. Deoxycholic acid acts as a detergent to solubilize fats for intestinal absorptio...
T0700 Ursodeoxycholic acid UDCA,Ursodiol Potassium Channel , Endogenous Metabolite
Ursodeoxycholic acid (UDCA) can be used to dissolve gallstones and reduce cholesterol absorption.
T2968 Hyodeoxycholic acid NSC 60672,α-Hyodeoxycholic Acid,HDCA FXR , Endogenous Metabolite , GPCR19
Hyodeoxycholic acid (NSC 60672) has been used in trials studying the treatment of Hypercholesterolemia.
T29078 Ursodeoxycholic acid sodium UDCA Na,UDCA sodium,Sodium Ursodeoxycholate,Ursodiol sodium,Ursodeoxycholic Acid (sodium salt),Ursodeoxycholate sodium FXR , Endogenous Metabolite , GPCR19
Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities. Ursodeoxycholic acid sodium acts as signaling molecule, exerting it...

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPH-01082 CMKLR1 Protein, Human, Recombinant (His) Human E. coli
CMKLR1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 45.1 kDa and the accession number is Q99788.
TMPJ-01304 C1QTNF1 Protein, Human, Recombinant (His) Human HEK293 Cells
C1QTNF1 is a secreted protein,contains 1 C1q domain and 1 collagen-like domain. C1qTNF proteins constitute a highly conserved family of Acrp30/Adiponectin paralogs that share a modular organization comprising an N-termin...
TMPH-03749 CYSLTR1 Protein, Human, Recombinant (His) Human E. coli
Receptor for cysteinyl leukotrienes mediating bronchoconstriction of individuals with and without asthma. Stimulation by LTD4 results in the contraction and proliferation of smooth muscle, edema, eosinophil migration and...
TMPH-03265 CMKLR2 Protein, Rat, Recombinant (His) Rat E. coli
Receptor for chemoattractant adipokine chemerin/RARRES2 suggesting a role for this receptor in the regulation of inflammation and energy homesotasis. Signals mainly via beta-arrestin pathway. Binding of RARRES2 activates...
TMPY-02837 GPR114 Protein, Human, Recombinant (hFc) Human HEK293 Cells
GPR114 belongs to the G-protein coupled receptor 2 family. Members of this family share a common molecular architecture which consists of seven transmembrane domains, three extracellular loops, three intracellular loops,...
TMPJ-00354 FZD1/Frizzled 1 Protein, Mouse, Recombinant (hFc) Mouse HEK293 Cells
Frizzled homolog 1 (FZD1), also known as Frizzled-1, a member of the G-protein-coupled receptor superfamily, mediates Wnt signaling by serving as a co-receptor with LRP-5 for Wnt ligands. The FZD1 protein contains a sign...
TMPY-02717 GPR37 Protein, Human, Recombinant (His) Human HEK293 Cells
GPR37 (cathepsin Z) is an orphan receptor that belongs to the G-protein coupled receptor 1 family. G protein-coupled receptors are a large protein family comprised of transmembrane receptors that sense molecules outside ...
TMPH-01385 GLP1R Protein, Human, Recombinant (His) Human HEK293 Cells
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ...
TMPK-01193 GPRC5D Protein-VLP, Mouse, Recombinant Mouse HEK293 Cells
Chimeric antigen receptor (CAR) T cells, a type of cell-based immunotherapy, have shown some promising results in multiple myeloma, a bone marrow cancer.The orphan G proteincoupled receptor, class C group 5 member D (GP...
TMPH-03301 GLP1R Protein, Rat, Recombinant (E. coli, His) Rat E. coli
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ...
TMPH-02676 GLP1R Protein, Mouse, Recombinant (His & SUMO) Mouse E. coli
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ...
TMPH-01384 GLP1R Protein, Human, Recombinant (E. coli, His) Human E. coli
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ...
TMPY-04562 GRK2 Protein, Human, Recombinant (His & GST) Human Baculovirus Insect Cells
G-protein coupled receptor kinase 2 (GRK2), also referred as Adrenergic, beta, receptor kinase 1 (ADRBK1), is a ubiquitous member of the G protein-coupled receptor kinase (GRK) family that appears to play a central, inte...
TMPJ-00983 ARRB1 Protein, Human, Recombinant (His) Human E. coli
β-Arrestin-1 (ARRB1) is a cytoplasmic protein that belongs to the arrestin family. ARRB1 is expressed at high levels in peripheral blood leukocytes and the central nervous system. ARRB1 regulates agonist-mediated G-prote...
TMPY-01165 FZD1/Frizzled 1 Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
Frizzled-1, also known as FZD1, belongs to theG-protein coupled receptor Fz/Smo family. FZD1 contains a signal peptide, a cysteine-rich domain in the N-terminal extracellular region, 7 transmembrane domains, and a C-term...
TMPY-02236 PTH1R Protein, Human, Recombinant (His) Human HEK293 Cells
Parathyroid hormone / parathyroid hormone-related peptide receptor, also known as PTH / PTHrP type I receptor, PTH/PTHr receptor, Parathyroid hormone 1 receptor, PTH1 receptor, PTH1R and PTHR, is a multi-pass membrane pr...
TMPY-02393 Thimet Oligopeptidase/THOP1 Protein, Mouse, Recombinant (His) Mouse Baculovirus Insect Cells
THOP1, also known as Thimet oligopeptidase 1, Thimet oligopeptidase, EC 3.4.24.15, or EP24.15, is a zinc(II) endopeptidase implicated in the processing of numerous physiological peptides. As an intracellular enzyme, high...
TMPY-04456 PKC nu Protein, Human, Recombinant (GST) Human Baculovirus Insect Cells
Serine/threonine-protein kinase D3, also known as Protein kinase C nu type, Protein kinase EPK2, PRKD3, EPK2 and PRKCN, is a cytoplasm and membrane protein that belongs to the protein kinase superfamily, CAMK Ser/Thr pro...
TMPY-04451 AMPK (G1/B1/A1) Heterotrimer Protein, Human, Recombinant (His & GST) Human Baculovirus Insect Cells
AMPK (G1/B1/A1) Heterotrimer Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 160 kDa and the accession number is P54619-1&Q9Y478-1&...
TMPY-03878 Integrin alpha V beta 6 Protein, Human, Recombinant (Flag & His) Human HEK293 Cells
Integrin alpha V beta 6 Protein, Human, Recombinant (Flag & His) is expressed in HEK293 mammalian cells with Flag and His tag. The predicted molecular weight is 190.4 kDa and the accession number is P06756-1&P18564-1.
TMPY-02501 CD3D & CD3E Heterodimer Protein, Human, Recombinant Human HEK293 Cells
CD3D & CD3E Heterodimer Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 77.5 kDa and the accession number is P04234-1&P07766-1.
TMPY-03745 CD3D & CD3E Heterodimer Protein, Human, Recombinant (Flag & His) Human HEK293 Cells
CD3D & CD3E Heterodimer Protein, Human, Recombinant (Flag & His) is expressed in HEK293 mammalian cells with Flag and His tag. The predicted molecular weight is 31.05 kDa and the accession number is P04234-1&P07766-1.
TMPY-03958 TGF alpha Protein, Human, Recombinant Human E. coli
The miR-137 served as a tumor suppressor in non-small cell lung cancer (NSCLC) and its suppressive effect is mediated by repressing TGFA expression. TGFA gene expression was significantly higher in tumor tissues compared...
TMPY-04069 Neurotrophin 3 Protein, Human, Recombinant Human E. coli
NTF3 (Neurotrophin 3) is a Protein Coding gene. The protein encoded by this gene is a member of the neurotrophin family, that controls the survival and differentiation of mammalian neurons. This protein is closely relate...
TMPY-02907 FGF-19 Protein, Human, Recombinant Human E. coli
FGF19, also known as FGF-19, is a member of the fibroblast growth factor (FGF) family. FGF family members possess broad mitogenic and cell survival activities, and are involved in a variety of biological processes, inclu...
TMPK-00383 ACE2/ACEH Protein, Human, Recombinant (His & Avi) Human HEK293 Cells
ACE2 (Angiotensin I Converting Enzyme 2) is a Protein Coding gene. Diseases associated with ACE2 include Severe Acute Respiratory Syndrome and Neurogenic Hypertension.The protein encoded by this gene belongs to the angio...
TMPY-01459 TNFR1/CD120a/TNFRSF1A Protein, Human, Recombinant (His) Human HEK293 Cells
TNFR1/CD120a/TNFRSF1A Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 22.7 kDa and the accession number is P19438-1.
TMPY-01827 CD30/TNFRSF8 Protein, Human, Recombinant (His) Human HEK293 Cells
CD30/TNFRSF8 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40 kDa and the accession number is P28908-1.
TMPY-01776 Carboxylesterase 2/CES2 Protein, Human, Recombinant (His) Human HEK293 Cells
Carboxylesterase 2/CES2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 60.4 kDa and the accession number is O00748-1.
TMPY-02019 CD59 Protein, Human, Recombinant (His) Human HEK293 Cells
CD59 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 10.2 kDa and the accession number is P13987-1.
TMPY-01461 EMAP-II/AIMP1 Protein, Human, Recombinant (His) Human E. coli
EMAP-II/AIMP1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 35 kDa and the accession number is Q12904-1.
TMPY-00972 FGFR2 Protein, Human, Recombinant (His & hFc) Human HEK293 Cells
FGFR2 Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 67.6 kDa and the accession number is P21802-1.
TMPY-01104 Coagulation factor XI/F11 Protein, Human, Recombinant (His) Human HEK293 Cells
Factor XI (plasma thromboplastin antecedent) is a plasma glycoprotein, and a zymogen acting as a serine protease which participates in blood coagulation as a catalyst in the conversion of factor IX to factor IXa in the p...
TMPY-01912 Cadherin 17/CDH17 Protein, Human, Recombinant (His) Human HEK293 Cells
Cadherin 17/CDH17 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 87 kDa and the accession number is Q12864-1.
TMPY-02031 B7-H3 Protein, Human, Recombinant (His) Human HEK293 Cells
B7-H3 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 48 kDa and the accession number is Q5ZPR3-1.
TMPY-02525 RGMA Protein, Human, Recombinant (His) Human HEK293 Cells
RGMa, also known as RGM domain family, member A, belongs to the RGM (repulsive guidance molecule) family whose members are membrane-associated glycoprotein. RGMa is a glycosylphosphatidylinositol-anchored glycoprotein th...
TMPY-04262 B7-H3 Protein, Human, Recombinant (His), Biotinylated Human HEK293 Cells
B7-H3 Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 48 kDa and the accession number is Q5ZPR3-1.
TMPY-00915 Serpin A1 Protein, Human, Recombinant (His) Human HEK293 Cells
Serpin A1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 45.7 kDa and the accession number is P01009-1.
TMPY-02836 MFGE8 Protein, Human, Recombinant (His) Human Baculovirus Insect Cells
MFGE8 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 42 kDa and the accession number is Q08431-1.
TMPY-01462 IL-11R alpha/IL-11RA Protein, Human, Recombinant (His) Human HEK293 Cells
IL-11R alpha/IL-11RA Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38.6 kDa and the accession number is Q14626-1.
TMPK-00176 BAFF/TNFSF13B Trimer Protein, Human, Recombinant (His & Flag) Human HEK293 Cells
B-cell activating factor (BAFF) also known as tumor necrosis factor ligand superfamily member 13B is a protein that in humans is encoded by the TNFSF13B gene.BAFF is a cytokine that belongs to the tumor necrosis factor (...
TMPY-02034 Siglec-2/CD22 Protein, Human, Recombinant (His) Human HEK293 Cells
Siglec-2/CD22 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.6 kDa and the accession number is P20273-1.
TMPY-02794 TLR2 Protein, Human, Recombinant (aa 1-587, His) Human Baculovirus Insect Cells
TLR2 Protein, Human, Recombinant (aa 1-587, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 65.5 kDa and the accession number is O60603-1.
TMPY-04799 IFNAR2 Protein, Human, Recombinant (His), Biotinylated Human HEK293 Cells
IFNAR2 Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.2 kDa and the accession number is P48551-1.
TMPY-02647 IFNAR1 Protein, Human, Recombinant (His) Human HEK293 Cells
IFNAR1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 48.6 kDa and the accession number is P17181-1.
TMPY-04826 LILRB5/CD85c Protein, Human, Recombinant (His) Human HEK293 Cells
A genetic variant in LILRB5 (leukocyte immunoglobulin-like receptor subfamily-B) (rs12975366: T > C: Asp247Gly) has been reported to be associated with lower creatine phosphokinase (CK) and lactate dehydrogenase (LDH) le...
TMPY-00740 SDF-1 Protein, Human, Recombinant (hFc) Human HEK293 Cells
SDF-1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 35.2 kDa and the accession number is P48061-1.
TMPY-04698 HER2/ERBB2 Protein, Human, Recombinant (aa 489-630, His) Human HEK293 Cells
HER2/ERBB2 Protein, Human, Recombinant (aa 489-630, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 17.1 kDa and the accession number is P04626-1.
TMPY-00203 LOXL2 Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
Lysyl oxidase homolog 2, also known as Lysyl oxidase-like protein 2, Lysyl oxidase-related protein 2, Lysyl oxidase-related protein WS9-14 and LOXL2, is a secreted protein that belongs to the lysyl oxidase family. LOXL2 ...
TMPK-00305 TGFBR1 Protein, Human, Recombinant (mFc & Avi) Human HEK293 Cells
transforming growth factor beta receptor 1 (TGFBR1), a key stimulator of tumor proliferation and metastasis, was a direct target of miR‑98‑5p. miR‑98‑5p overexpression resulted in the downregulation of TGFBR1 and the sup...
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CMKLR1 Protein, Human, Recombinant (His)
TMPH-01082
Species: Human
Expression System: E. coli
C1QTNF1 Protein, Human, Recombinant (His)
TMPJ-01304
Species: Human
Expression System: HEK293 Cells
CYSLTR1 Protein, Human, Recombinant (His)
TMPH-03749
Species: Human
Expression System: E. coli
CMKLR2 Protein, Rat, Recombinant (His)
TMPH-03265
Species: Rat
Expression System: E. coli
GPR114 Protein, Human, Recombinant (hFc)
TMPY-02837
Species: Human
Expression System: HEK293 Cells
FZD1/Frizzled 1 Protein, Mouse, Recombinant (hFc)
TMPJ-00354
Species: Mouse
Expression System: HEK293 Cells
GPR37 Protein, Human, Recombinant (His)
TMPY-02717
Species: Human
Expression System: HEK293 Cells
GLP1R Protein, Human, Recombinant (His)
TMPH-01385
Species: Human
Expression System: HEK293 Cells
GPRC5D Protein-VLP, Mouse, Recombinant
TMPK-01193
Species: Mouse
Expression System: HEK293 Cells
GLP1R Protein, Rat, Recombinant (E. coli, His)
TMPH-03301
Species: Rat
Expression System: E. coli
GLP1R Protein, Mouse, Recombinant (His & SUMO)
TMPH-02676
Species: Mouse
Expression System: E. coli
GLP1R Protein, Human, Recombinant (E. coli, His)
TMPH-01384
Species: Human
Expression System: E. coli
GRK2 Protein, Human, Recombinant (His & GST)
TMPY-04562
Species: Human
Expression System: Baculovirus Insect Cells
ARRB1 Protein, Human, Recombinant (His)
TMPJ-00983
Species: Human
Expression System: E. coli
FZD1/Frizzled 1 Protein, Mouse, Recombinant (His)
TMPY-01165
Species: Mouse
Expression System: HEK293 Cells
PTH1R Protein, Human, Recombinant (His)
TMPY-02236
Species: Human
Expression System: HEK293 Cells
Thimet Oligopeptidase/THOP1 Protein, Mouse, Recombinant (His)
TMPY-02393
Species: Mouse
Expression System: Baculovirus Insect Cells
PKC nu Protein, Human, Recombinant (GST)
TMPY-04456
Species: Human
Expression System: Baculovirus Insect Cells
AMPK (G1/B1/A1) Heterotrimer Protein, Human, Recombinant (His & GST)
TMPY-04451
Species: Human
Expression System: Baculovirus Insect Cells
Integrin alpha V beta 6 Protein, Human, Recombinant (Flag & His)
TMPY-03878
Species: Human
Expression System: HEK293 Cells
CD3D & CD3E Heterodimer Protein, Human, Recombinant
TMPY-02501
Species: Human
Expression System: HEK293 Cells
CD3D & CD3E Heterodimer Protein, Human, Recombinant (Flag & His)
TMPY-03745
Species: Human
Expression System: HEK293 Cells
TGF alpha Protein, Human, Recombinant
TMPY-03958
Species: Human
Expression System: E. coli
Neurotrophin 3 Protein, Human, Recombinant
TMPY-04069
Species: Human
Expression System: E. coli
FGF-19 Protein, Human, Recombinant
TMPY-02907
Species: Human
Expression System: E. coli
ACE2/ACEH Protein, Human, Recombinant (His & Avi)
TMPK-00383
Species: Human
Expression System: HEK293 Cells
TNFR1/CD120a/TNFRSF1A Protein, Human, Recombinant (His)
TMPY-01459
Species: Human
Expression System: HEK293 Cells
CD30/TNFRSF8 Protein, Human, Recombinant (His)
TMPY-01827
Species: Human
Expression System: HEK293 Cells
Carboxylesterase 2/CES2 Protein, Human, Recombinant (His)
TMPY-01776
Species: Human
Expression System: HEK293 Cells
CD59 Protein, Human, Recombinant (His)
TMPY-02019
Species: Human
Expression System: HEK293 Cells
EMAP-II/AIMP1 Protein, Human, Recombinant (His)
TMPY-01461
Species: Human
Expression System: E. coli
FGFR2 Protein, Human, Recombinant (His & hFc)
TMPY-00972
Species: Human
Expression System: HEK293 Cells
Coagulation factor XI/F11 Protein, Human, Recombinant (His)
TMPY-01104
Species: Human
Expression System: HEK293 Cells
Cadherin 17/CDH17 Protein, Human, Recombinant (His)
TMPY-01912
Species: Human
Expression System: HEK293 Cells
B7-H3 Protein, Human, Recombinant (His)
TMPY-02031
Species: Human
Expression System: HEK293 Cells
RGMA Protein, Human, Recombinant (His)
TMPY-02525
Species: Human
Expression System: HEK293 Cells
B7-H3 Protein, Human, Recombinant (His), Biotinylated
TMPY-04262
Species: Human
Expression System: HEK293 Cells
Serpin A1 Protein, Human, Recombinant (His)
TMPY-00915
Species: Human
Expression System: HEK293 Cells
MFGE8 Protein, Human, Recombinant (His)
TMPY-02836
Species: Human
Expression System: Baculovirus Insect Cells
IL-11R alpha/IL-11RA Protein, Human, Recombinant (His)
TMPY-01462
Species: Human
Expression System: HEK293 Cells
BAFF/TNFSF13B Trimer Protein, Human, Recombinant (His & Flag)
TMPK-00176
Species: Human
Expression System: HEK293 Cells
Siglec-2/CD22 Protein, Human, Recombinant (His)
TMPY-02034
Species: Human
Expression System: HEK293 Cells
TLR2 Protein, Human, Recombinant (aa 1-587, His)
TMPY-02794
Species: Human
Expression System: Baculovirus Insect Cells
IFNAR2 Protein, Human, Recombinant (His), Biotinylated
TMPY-04799
Species: Human
Expression System: HEK293 Cells
IFNAR1 Protein, Human, Recombinant (His)
TMPY-02647
Species: Human
Expression System: HEK293 Cells
LILRB5/CD85c Protein, Human, Recombinant (His)
TMPY-04826
Species: Human
Expression System: HEK293 Cells
SDF-1 Protein, Human, Recombinant (hFc)
TMPY-00740
Species: Human
Expression System: HEK293 Cells
HER2/ERBB2 Protein, Human, Recombinant (aa 489-630, His)
TMPY-04698
Species: Human
Expression System: HEK293 Cells
LOXL2 Protein, Mouse, Recombinant (His)
TMPY-00203
Species: Mouse
Expression System: HEK293 Cells
TGFBR1 Protein, Human, Recombinant (mFc & Avi)
TMPK-00305
Species: Human
Expression System: HEK293 Cells
Cat No. Product Name
L7600 Chemokine Inhibitor Library

59 compounds
A unique collection of 59 chemokines or chemokine receptors targeted compounds for high throughput and high content screening;
TargetMol